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Pseudopolymorphic Forms Of A Hiv Protease Inhibitor - EP2767539

The patent EP2767539 was granted to Janssen R&D Ireland on Jul 12, 2017. The application was originally filed on May 16, 2003 under application number EP14168686A. The patent is currently recorded with a legal status of "Opposition Rejected".

EP2767539

JANSSEN R&D IRELAND
Application Number
EP14168686A
Filing Date
May 16, 2003
Status
Opposition Rejected
Feb 10, 2023
Grant Date
Jul 12, 2017
External Links
Slate, Register, Google Patents

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COOKEApr 12, 2018ELKINGTON AND FIFEADMISSIBLE

Patent Citations (9) New

Patent citations refer to prior patents cited during different phases such as opposition or international search.

Citation PhasePublication NumberPublication Link
DESCRIPTIONEP0715618
DESCRIPTIONUS6248775
DESCRIPTIONWO9967417
OPPOSITIONUS6248775
OPPOSITIONWO03106461
OPPOSITIONWO9506030
OPPOSITIONWO9967417
SEARCHWO9506030
SEARCHWO9967417

Non-Patent Literature (NPL) Citations (14) New

NPL citations refer to non-patent references such as research papers, articles, or other publications cited during examination or opposition phases.

Citation PhaseReference TextLink
DESCRIPTION- BIOORGANIC AND CHEMIST LETTERS, (1998), vol. 8, pages 687 - 690-
OPPOSITION- Aulton, Pharmaceutics: The Science of Dosage Form Design, (20020000), pages 144 - 146 , 239-
OPPOSITION- BORKA L et al., "Crystal polymorphism of pharmaceuticals", Acta Pharmaceutica, (19900000), vol. 40, pages 71 - 94, XP009031944-
OPPOSITION- BYRN S R et al., "Solid-State Chemistry of Drugs", Solid-State Chemistry Of Drugs, vol. 12, pages 82 - 85, XP002588305-
OPPOSITION- GIRON et al., "Thermal analysis and calorimetric methods in the characterisation of polymorphs and solvates", Thermochimica acta, (19950000), vol. 248, pages 1 - 59, XP002101808
OPPOSITION- GRUNENBERG A. et al., "Theoretical derivation and practical application of energy/temperature diagrams as an instrument in preformulation studies of polymorphic drug substances", International Journal of Pharmaceutics, (19960308), vol. 129, pages 147 - 158, XP000909867
OPPOSITION- GHOSH A K et al., "Potent HIV protease inhibitors incorporating high-affinity P2-ligands and (R)-(hydroxyethylamino) sulfonamide isostere", Bioorganic & Medicinal Chemistry Letters, vol. 8, no. 6, pages 687 - 690, XP004136945
OPPOSITION- GHOSH A K et al., "Nonpeptidal P2 Ligands for HIV protease Inhibitors: Structure-Based Design Synthesis and Biological Evaluation", Journal Of Medicinal Chemistry, vol. 39, pages 3278 - 3290, XP002193358
SEARCH- BORKA L ET AL, "Crystal polymorphism of pharmaceuticals", ACTA PHARMACEUTICA JUGOSLAVICA, SAVEZ FARMACEUTSKIH DRUSTAVA JUGOSLAVIJE, ZAGREB, YU, (1990), vol. 40, ISSN 0001-6667, pages 71 - 94, XP002195530 [Y] 1-17 * the whole document *-
SEARCH- BYRN S R ET AL, Solid-State Chemistry of Drugs, SOLID-STATE CHEMISTRY OF DRUGS, SSCI INC, WEST LAFAYETTE, PAGE(S) 82 - 85, (19990110), ISBN 978-0-9670671-0-0, XP002588305 [Y] 1-17 * the whole document *-
SEARCH- GIRON ET AL, "Thermal analysis and calorimetric methods in the characterisation of polymorphs and solvates", THERMOCHIMICA ACTA, ELSEVIER SCIENCE PUBLISHERS, AMSTERDAM, NL, (1995), vol. 248, ISSN 0040-6031, pages 1 - 59, XP002101808 [Y] 1-17 * the whole document *
SEARCH- GRUNENBERG A ET AL, "THEORETICAL DERIVATION AND PRACTICAL APPLICATION OF ENERGY/TEMPERATURE DIAGRAMS AS AN INSTRUMENT IN PREFORMULATION STUDIES OF POLYMORPHIC DRUG SUBSTANCES", INTERNATIONAL JOURNAL OF PHARMACEUTICS, AMSTERDAM, NL, (19960308), vol. 129, ISSN 0378-5173, pages 147 - 158, XP000909867 [Y] 1-17 * the whole document *
SEARCH- GHOSH A K ET AL, "Potent HIV protease inhibitors incorporating high-affinity P2-ligands and (R)-(hydroxyethylamino)sulfonamide isostere", BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, OXFORD, GB, (19980317), vol. 8, no. 6, ISSN 0960-894X, pages 687 - 690, XP004136945 [YD] 1-17 * the whole document *
SEARCH- GHOSH A K ET AL, "Nonpeptidal P2 Ligands for HIV protease Inhibitores: Structure-Based Design Synthesis and Biological Evaluation", JOURNAL OF MEDICINAL CHEMISTRY, AMERICAN CHEMICAL SOCIETY, US, (19960816), vol. 39, doi:10.1021/JM960128K, ISSN 0022-2623, pages 3278 - 3290, XP002193358 [Y] 1-17 * the whole document * * see p.3281, Table 1 *

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