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The patent EP3078667 was granted to The United States OF America on Nov 21, 2018. The application was filed on Jan 25, 2002 under application number EP16157001A. The patent is currently recorded with a legal status of "Granted And Under Opposition".
Stable, pharmaceutically acceptable compositions of boronic acid compounds are prepared by lyophilizing an aqueous mixture of the boronic acid and a dihydroxy compound, such as mannitol. The resulting lyophilized composition readily releases the boronic acid compound upon dissolution in aqueous media, forming a boronate ester that equilibrates with the free boronic acid. The compositions exhibit enhanced stability and longer shelf life compared to free boronic acid compounds, and can be reconstituted to provide a bioactive boronic acid compound.

Patent oppositions filed by competitors challenge the validity of a granted patent. These oppositions are typically based on claims of prior art, lack of novelty, or non-obviousness. They are a key part of the process for determining a patent's strength and enforceability.
| Company | Opposition Date | Representative | Opposition Status |
|---|---|---|---|
| GENERICS UK | Aug 21, 2019 | ELKINGTON AND FIFE | ADMISSIBLE |
| ACCORD HEALTHCARE | Aug 20, 2019 | TER MEER STEINMEISTER & PARTNER | ADMISSIBLE |
| DR REDDYS LABORATORIES BETAPHARM ARZNEIMITTEL | Aug 20, 2019 | HOPFNER | ADMISSIBLE |
| ZENTIVA KS | Aug 20, 2019 | BIRD & BIRD | ADMISSIBLE |
| KRKA | Aug 20, 2019 | KUTZENBERGER WOLFF & PARTNER | WITHDRAWN |
| PENTAFARMA | Aug 19, 2019 | KUTZENBERGER WOLFF & PARTNER | ADMISSIBLE |
| SYNTHON | Aug 16, 2019 | - | ADMISSIBLE |
| LEK PHARMACEUTICALS DD | Aug 14, 2019 | KRAUS & LEDERER PARTGMBB | WITHDRAWN |
| PFIZER | Aug 7, 2019 | ELKINGTON AND FIFE | ADMISSIBLE |
| FRESENIUS KABI DEUTSCHLAND | Jun 17, 2019 | FRESENIUS KABI DEUTSCHLAND | ADMISSIBLE |
| TEVA PHARMACEUTICALS | May 29, 2019 | GRAF VON STOSCH PATENTANWALTSGESELLSCHAFT | ADMISSIBLE |
Patent citations refer to prior patents cited during different phases such as opposition or international search.
| Citation Phase | Publication Number |
|---|---|
| DESCRIPTION | US4499082 |
| DESCRIPTION | US5106948 |
| DESCRIPTION | US5169841 |
| DESCRIPTION | US5187157 |
| DESCRIPTION | US5242904 |
| DESCRIPTION | US5250720 |
| DESCRIPTION | US5780454 |
| DESCRIPTION | US6066730 |
| DESCRIPTION | US6083903 |
| DESCRIPTION | US6297217 |
| DESCRIPTION | WO9835691 |
| DESCRIPTION | WO9915183 |
| OPPOSITION | EP0308238 |
| OPPOSITION | EP1355910 |
| OPPOSITION | EP2251344 |
| OPPOSITION | EP3078667 |
| OPPOSITION | US4360694 |
| OPPOSITION | US4670262 |
| OPPOSITION | US5505953 |
| OPPOSITION | US5536735 |
| OPPOSITION | US5780454 |
| OPPOSITION | US5935994 |
| OPPOSITION | US5962049 |
| OPPOSITION | US5985842 |
| OPPOSITION | US6066730 |
| OPPOSITION | US6083903 |
| OPPOSITION | WO0057887 |
| OPPOSITION | WO02059130 |
| OPPOSITION | WO9613266 |
| OTHER | EP1355910 |
| OTHER | EP2251344 |
| SEARCH | WO9613266 |
The dossier documents provide a comprehensive record of the patent's prosecution history - including filings, correspondence, and decisions made by patent offices - and are crucial for understanding the patent's legal journey and any challenges it may have faced during examination.
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Decision to grant a European patent
Search/Exam
Oct 5, 2018
(Electronic) Receipt
Search/Exam
Oct 5, 2018
Oct 5, 2018
Oct 5, 2018
Oct 5, 2018
Filing of the translations of the claims
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Oct 5, 2018
Intention to grant (signatures)
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Oct 5, 2018
Letter accompanying subsequently filed items
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Oct 5, 2018
Text intended for grant (clean copy)
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Oct 5, 2018
Sep 21, 2018
Sep 5, 2018
Aug 31, 2018
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Aug 29, 2018
Non-patent literature filed by a third party
Search/Exam
Aug 29, 2018
Non-patent literature filed by a third party
Search/Exam
Aug 29, 2018
Non-patent literature filed by a third party
Search/Exam
Aug 29, 2018
Non-patent literature filed by a third party
Search/Exam
Aug 29, 2018
Non-patent literature filed by a third party
Search/Exam
Aug 29, 2018
Non-patent literature filed by a third party
Search/Exam
Aug 29, 2018
Non-patent literature filed by a third party
Search/Exam
Aug 29, 2018
Non-patent literature filed by a third party
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Aug 29, 2018
Non-patent literature filed by a third party
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Aug 29, 2018
Observations by third parties
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Aug 27, 2018
(Electronic) Receipt
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Aug 27, 2018
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Aug 27, 2018
Non-patent literature filed by a third party
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Aug 27, 2018
Non-patent literature filed by a third party
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Aug 27, 2018
Non-patent literature filed by a third party
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Aug 27, 2018
Non-patent literature filed by a third party
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Aug 27, 2018
Non-patent literature filed by a third party
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Aug 27, 2018
Observations by third parties
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Aug 23, 2018
(Electronic) Receipt
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Aug 23, 2018
Filing of the translations of the claims
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Aug 23, 2018
French translation of claims
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Aug 23, 2018
German translation of the claims
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Aug 23, 2018
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Aug 22, 2018
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Aug 22, 2018
Intention to grant (signatures)
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Aug 22, 2018
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Aug 22, 2018
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Aug 6, 2018
Non-patent literature filed by a third party
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Aug 6, 2018
Non-patent literature filed by a third party
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Aug 6, 2018
Observations by third parties
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Jun 29, 2018
(Electronic) Receipt
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Jun 29, 2018
Amended claims with annotations
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Jun 29, 2018
Amended claims with annotations
Search/Exam
Jun 29, 2018
Claims
Search/Exam
Jun 29, 2018
Claims
Search/Exam
Jun 29, 2018
Letter accompanying subsequently filed items
Search/Exam
Jun 29, 2018
Jun 6, 2018
Annex to the communication
Search/Exam
Jun 6, 2018
Communication from the Examining Division
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May 24, 2018
(Electronic) Receipt
Search/Exam
May 24, 2018
Amended claims with annotations
Search/Exam
May 24, 2018
Amended claims with annotations
Search/Exam
May 24, 2018
Amended claims with annotations
Search/Exam
May 24, 2018
Amended claims with annotations
Search/Exam
May 24, 2018
Amended claims with annotations
Search/Exam
May 24, 2018
Amended claims with annotations
Search/Exam
May 24, 2018
Citation for the examination procedure
Search/Exam
May 24, 2018
Citation for the examination procedure
Search/Exam
May 24, 2018
Claims
Search/Exam
May 24, 2018
Claims
Search/Exam
May 24, 2018
Claims
Search/Exam
May 24, 2018
Claims
Search/Exam
May 24, 2018
Claims
Search/Exam
May 24, 2018
Claims
Search/Exam
May 24, 2018
Letter accompanying subsequently filed items
Search/Exam
May 24, 2018
May 16, 2018
May 9, 2018
Feb 20, 2018
Annex to the communication
Search/Exam
Feb 20, 2018
Communication from the Examining Division
Search/Exam
Feb 14, 2018
Refund of fees
Search/Exam
Feb 9, 2018
(Electronic) Receipt
Search/Exam
Feb 9, 2018
Citation filed by a third party
Search/Exam
Feb 9, 2018
Letter accompanying subsequently filed items
Search/Exam
Feb 9, 2018
Non-patent literature filed by a third party
Search/Exam
Feb 9, 2018
Observations by third parties
Search/Exam
Feb 9, 2018
Observations by third parties
Search/Exam
Feb 9, 2018
Observations by third parties
Search/Exam
Jan 31, 2018
Jan 31, 2018
Jan 31, 2018
Jan 25, 2018
(Electronic) Receipt
Search/Exam
Jan 25, 2018
Letter accompanying subsequently filed items
Search/Exam
Jan 25, 2018
Non-patent literature filed by a third party
Search/Exam
Jan 25, 2018
Observations by third parties
Search/Exam
Jan 25, 2018
Patent document filed by a Third party
Search/Exam
Jan 25, 2018
Patent document filed by a Third party
Search/Exam
Jan 23, 2018
Letter accompanying subsequently filed items
Search/Exam
Jan 23, 2018
Non-patent literature filed by a third party
Search/Exam
Jan 23, 2018
Patent document filed by a Third party
Search/Exam
Jan 2, 2018
(Electronic) Receipt
Search/Exam
Jan 2, 2018
Jan 2, 2018
Jan 2, 2018
Filing of the translations of the claims
Search/Exam
Jan 2, 2018
French translation of claims
Search/Exam
Jan 2, 2018
German translation of the claims
Search/Exam
Jan 2, 2018
Intention to grant (signatures)
Search/Exam
Jan 2, 2018
Letter accompanying subsequently filed items
Search/Exam
Jan 2, 2018
Text intended for grant (clean copy)
Search/Exam
Jan 2, 2018
Nov 13, 2017
Examination started
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Jul 31, 2017
Decision to allow further processing
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Jul 21, 2017
(Electronic) Receipt
Search/Exam
Jul 21, 2017
Jul 21, 2017
Amended claims with annotations
Search/Exam
Jul 21, 2017
Jul 21, 2017
Amended description with annotations
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Jul 21, 2017
Letter accompanying subsequently filed items
Search/Exam
Jul 21, 2017
Request for further processing
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May 22, 2017
Apr 5, 2017
(Electronic) Receipt
Search/Exam
Apr 5, 2017
Letter accompanying subsequently filed items
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Apr 5, 2017
Letter concerning fees and payments
Search/Exam
Oct 17, 2016
Sep 14, 2016
Notification of forthcoming publication
Search/Exam
Jul 13, 2016
Refund of fees
Search/Exam
Jul 1, 2016
Jul 1, 2016
European search opinion
Search/Exam
Jul 1, 2016
European search report
Search/Exam
Jul 1, 2016
Information on Search Strategy
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Jun 17, 2016
Search started
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(Electronic) Receipt
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May 26, 2016
Claims
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May 26, 2016
Letter accompanying subsequently filed items
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May 26, 2016
Matter concerning the application
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Apr 15, 2016
Communication to designated inventor
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Mar 16, 2016
Invitation to file claims
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Feb 23, 2016
Abstract
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Feb 23, 2016
Feb 23, 2016
Annex
Search/Exam
Feb 23, 2016
Description
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Feb 23, 2016
Designation of inventor
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Feb 23, 2016
Matter concerning the application
Search/Exam
Feb 23, 2016
Request for grant of a European patent
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Feb 23, 2016
Submission concerning representation
Search/Exam
Aug 7, 2002