| OPPOSITION | - Natasha Thorne, Min Shen, Wendy a. Lea, Anton Simeonov, Scott Lovell, Douglas s. Auld, James Inglese, "Firefly Luciferase in Chemical Biology: A Compendium of Inhibitors, Mechanistic Evaluation of Chemotypes, and Suggested Use As a Reporter", Chemistry & Biology, CURRENT BIOLOGY, LONDON, GB, GB , (20120801), vol. 19, no. 8, doi:10.1016/j.chembiol.2012.07.015, ISSN 1074-5521, pages 1060 - 1072, XP055373470 | |
| OPPOSITION | - Rozbeh Jafari, Helena Almqvist, Hanna Axelsson, Marina Ignatushchenko, Thomas Lundbäck, Pär Nordlund, Daniel Martinez Molina, "The cellular thermal shift assay for evaluating drug target interactions in cells", Nature Protocols, vol. 9, no. 9, doi:10.1038/nprot.2014.138, ISSN 17542189, pages 2100 - 2122, XP055193929 | |
| OPPOSITION | - Rehmann Holger, "Epac-Inhibitors: Facts and Artefacts", Scientific reports, Nature Publishing Group, US, US , (20131001), vol. 3, no. 1, doi:10.1038/srep03032, ISSN 2045-2322, page 3032, XP093297441 | |
| OPPOSITION | - Daniel Martinez Molina, Jafari R; Ignatushchenko M; Seki T; Larsson E A; Dan C; Sreekumar L; Cao Y; Nordlund P, "Monitoring drug target engagement in cells and tissues using the cellular thermal shift assay", Science - Author Manuscript, American Association for the Advancement of Science, US, US , (20130705), vol. 341, no. 6141, doi:10.1126/science.1233606, ISSN 0036-8075, pages 84 - 87, XP055471723 | |
| OPPOSITION | - Krishna Sankar N., Luan Chi-Hao, Mishra Rama K., Xu Li, Scheidt Karl A., Anderson Wayne F., Bergan Raymond C., "A Fluorescence-Based Thermal Shift Assay Identifies Inhibitors of Mitogen Activated Protein Kinase Kinase 4", PLOS ONE, Public Library of Science, US, US , (20131201), vol. 8, no. 12, doi:10.1371/journal.pone.0081504, ISSN 1932-6203, page e81504, XP093297437 | |
| SEARCH | - MELANIE L. DART ET AL, "Homogeneous Assay for Target Engagement Utilizing Bioluminescent Thermal Shift", ACS MEDICINAL CHEMISTRY LETTERS, (20180419), doi:10.1021/acsmedchemlett.8b00081, ISSN 1948-5875, XP055475102 [T] * the whole document * | |
| SEARCH | - MATTHEW B. ROBERS ET AL, "Target engagement and drug residence time can be observed in living cells with BRET", NATURE COMMUNICATIONS, (20151203), vol. 6, doi:10.1038/ncomms10091, page 10091, XP055271302 [AP] 1-23 * the whole document * | |
| SEARCH | - ROZBEH JAFARI ET AL, "The cellular thermal shift assay for evaluating drug target interactions in cells", NATURE PROTOCOLS, (20140807), vol. 9, no. 9, doi:10.1038/nprot.2014.138, ISSN 1754-2189, pages 2100 - 2122, XP055193929 [A] 1-23 * the whole document * | |
| SEARCH | - DANIEL MARTINEZ MOLINA ET AL, "Monitoring drug target engagement in cells and tissues using the cellular thermal shift assay", SCIENCE, US, (20130523), vol. 341, no. 6141, doi:10.1126/science.1233606, ISSN 0036-8075, pages 84 - 87, XP055471723 [A] 1-23 * the whole document * | |