| OPPOSITION | - Dave A. Miller; Marco Gil , " Chapter 10 Spray-Drying Technology", Formulating Poorly Water-Soluble Drugs, Springer, (20111203), pages 363 - 442, doi:10.1007/978-1-4614-1144-4_10, XP009556892 | |
| OPPOSITION | - Justin R. Hughey, Robert O. Williams III , "Chapter 3 Solid-State Techniques for Improving Solubility", Formulating Poorly Water-Soluble Drugs, Springer , (20111203), pages 95 - 131, doi:10.1007/978-1-4614-1144-4_3, ISBN 978-1-4614-1143-7, XP009556890 | |
| OPPOSITION | - Navnit Shah, Harpreet Sandhu, Duk Soon Choi, Oskar Kalb, Susanne Page, Nicole Wyttenbach , "Chapter 8 Structured Development Approach for Amorphous Systems", Formulating Poorly Water-Soluble Drugs, Springer , (20111203), pages 267 - 310, doi:10.1007/978-1-4614-1144-4_8, ISBN 978-1-4614-1143-7, XP009556891 | |
| OPPOSITION | - Bryan D. Smith, Michael D. Kaufman, Wei-Ping Lu, Anu Gupta, Cynthia B. Leary, Scott C. Wise, Thomas J. Rutkoski, Yu Mi Ahn, Gada Al-Ani, Stacie L. Bulfer, Timothy M. Caldwell, Lawrence Chun, Carol L. Ensinger, Molly M. Hood, Arin Mckinley, William C. Patt, Rodrigo Ruiz-Soto, Ying Su, Hanumaiah Telikepalli, Ajia Town, Benjamin A. Turner, Lakshminarayana Vogeti, Subha Vogeti, Karen Yates, Filip Janku, Albiruni Ryan Abdul Razak, Oliver Rosen, Michael C. Heinrich, Daniel L. Flynn, "Ripretinib (DCC-2618) Is a Switch Control Kinase Inhibitor of a Broad Spectrum of Oncogenic and Drug-Resistant KIT and PDGFRA Variants", CANCER CELL, CELL PRESS, US, US , (20190501), vol. 35, no. 5, doi:10.1016/j.ccell.2019.04.006, ISSN 1535-6108, pages 738 - 751.e9, XP055738739 | |
| OPPOSITION | - Konno, H. ; Handa, T. ; Alonzo, D.E. ; Taylor, L.S., "Effect of polymer type on the dissolution profile of amorphous solid dispersions containing felodipine", European journal of pharmaceutics and biopharmaceutics, ELSEVIER SCIENCE PUBLISHERS B.V., AMSTERDAM., NL, NL , (20081001), vol. 70, no. 2, doi:10.1016/j.ejpb.2008.05.023, ISSN 0939-6411, pages 493 - 499, XP025470891 | |
| OPPOSITION | - Miller Jonathan M., Beig Avital, Carr Robert A., Spence Julie K., Dahan Arik, "A Win-Win Solution in Oral Delivery of Lipophilic Drugs: Supersaturation via Amorphous Solid Dispersions Increases Apparent Solubility without Sacrifice of Intestinal Membrane Permeability", Molecular Pharmaceutics, American Chemical Society, US, US , (20120702), vol. 9, no. 7, doi:10.1021/mp300104s, ISSN 1543-8384, pages 2009 - 2016, XP055812634 | |
| OPPOSITION | - Tanno Fumié; Nishiyama Yuichi; Kokubo Hiroyasu; Obara Sakaé, "Evaluation of hypromellose acetate succinate (HPMCAS) as a carrier in solid dispersions.", Journal Drug Development and Industrial Pharmacy, NEW YORK, NY, US, US , (20040101), vol. 30, no. 1, doi:10.1081/DDC-120027506, ISSN 0363-9045, pages 9 - 17, XP009124621 | |
| OPPOSITION | - Nemunaitis John, Bauer Sebastian, Blay Jean-Yves, Choucair Khalil, Gelderblom Hans, George Suzanne, Schöffski Patrick, Mehren Margaret Von, Zalcberg John, Achour Haroun, Ruiz-Soto Rodrigo, Heinrich Michael C, "Intrigue: Phase III Study of Ripretinib Versus Sunitinib in Advanced Gastrointestinal Stromal Tumor After Imatinib", FUTURE ONCOLOGY, FUTURE MEDICINE LTD., LONDON, GB, GB , (20200131), vol. 16, no. 1, doi:10.2217/fon-2019-0633, ISSN 1479-6694, pages 4251 - 4264, XP093202201 | |
| OPPOSITION | - Dallas B. Warren, Benameur Hassan, Porter Christopher J.H., Pouton Colin W., "Using polymeric precipitation inhibitors to improve the absorption of poorly water-soluble drugs: A mechanistic basis for utility", Journal of Drug Targeting, (20101201), vol. 18, no. 10, doi:10.3109/1061186X.2010.525652, ISSN 1061186X, pages 704 - 731, XP055027752 | |