Patent No. EP2299987 (titled "Capsule Pharmaceutical Dosage Form Comprising A Suspension Formulation Of An Indolinone Derivative") was filed by Boehringer Ingelheim on Jun 4, 2009. The application was issued on Feb 21, 2018.
Active substance 3-Z-[1-(4-(N-((4-methyl-piperazin-1-yl)-methylcarbonyl)-N-methyl-amino)-anilino)-1-phenyl-methylene]-6-methoxycarbonyl-2-indolinone-monoethanesulphonate. The active substance includes a lipid suspension containing a viscous suspension of 3-Z-[1-(4-(N-((4-methyl-piperazin-1-yl)-methylcarbonyl)-N-methyl-amino)-anilino)-1-phenyl-methylene]-6-methoxycarbonyl-2-indolinone-monoethanesulphonate, which is based on a lipid suspension formulation.

Patent oppositions filed by competitors challenge the validity of a granted patent. These oppositions are typically based on claims of prior art, lack of novelty, or non-obviousness. They are a key part of the process for determining a patent's strength and enforceability.
| Company | Opposition Date | Representative |
|---|---|---|
| GALENICUM HEALTH SLU | Nov 21, 2018 | GALENICUM HEALTH SLU |
| GENERICS UK | Nov 21, 2018 | TER MEER STEINMEISTER & PARTNER |
| TEVA PHARMACEUTICALS | Nov 21, 2018 | KRAUS & LEDERER PARTGMBB |
| ZENTIVA GROUP | Nov 21, 2018 | GREINER |
The dossier documents provide a comprehensive record of the patent's prosecution history - including filings, correspondence, and decisions made by patent offices - and are crucial for understanding the patent's legal journey and any challenges it may have faced during examination.
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