Patent No. EP3488857 (titled "Compositions Of Glp-1 Peptides And Preparation Thereof") was filed by Novo Nordisk on Mar 15, 2013. The application was issued on Oct 4, 2023.
Improving oral delivery of GLP-1 peptides like glucagon-like peptide-1 (GLP-1) for treating diabetes and obesity. The invention involves designing granules for tablet formulations containing GLP-1 peptides and delivery agents like SNAC. The granules are prepared by mixing the peptide, fillers, and binders, then the delivery agent mix. This two-step granulation process allows separate optimization of peptide and delivery properties. The resulting granules have improved dissolution profiles for faster GLP-1 release compared to co-granulating.

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| Company | Opposition Date | Representative |
|---|---|---|
| GENERICS UK | Mar 7, 2024 | TER MEER STEINMEISTER & PARTNER |
| HAMM & WITTKOPP | Mar 7, 2024 | HAMM & WITTKOPP |
| HEXAL | Mar 7, 2024 | MAIWALD |
| POLPHARMA | Mar 7, 2024 | MAIWALD |
| STRAWMAN | Mar 5, 2024 | HOFFMANN EITLE |
The dossier documents provide a comprehensive record of the patent's prosecution history - including filings, correspondence, and decisions made by patent offices - and are crucial for understanding the patent's legal journey and any challenges it may have faced during examination.
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