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The patent EP3524595 was granted to Eisai R&D Management on Aug 10, 2022. The application was filed on Aug 26, 2015 under application number EP19151846A. The patent is currently recorded with a legal status of "Granted And Under Opposition".
Quinline derivative that is easy to remove such impurities by a common purification method such as chromatography and crystallization. The derivative comprises a compound represented by formula (IV) or a salt thereof; an organometallic reagent such as butyllithium, methyllithium, lithium bistrimethylsilylamide, sodium bistrimethylsilylamide or potassium bistrimethylsilylamide; a hydride such as lithium hydride, sodium hydride or potassium hydride; a heterocyclic compound such as imidazole, pyridine, dimethylpyridine, trimethylpyridine or 4-dimethylaminopyridine; or an organic amine such as triethylamine, N,N-diisopropylethylamine or diazabicycloundecene.

Patent oppositions filed by competitors challenge the validity of a granted patent. These oppositions are typically based on claims of prior art, lack of novelty, or non-obviousness. They are a key part of the process for determining a patent's strength and enforceability.
| Company | Opposition Date | Representative | Opposition Status |
|---|---|---|---|
| ACCORD HEALTHCARE | May 10, 2023 | UEXKULL & STOLBERG | ADMISSIBLE |
| AECHTER | May 10, 2023 | TER MEER STEINMEISTER & PARTNER | ADMISSIBLE |
| GENERICS UK | May 10, 2023 | RUSSELL | ADMISSIBLE |
| MAIWALD | May 10, 2023 | MAIWALD | ADMISSIBLE |
| STADA ARZNEIMITTEL | May 10, 2023 | HAMM & WITTKOPP | ADMISSIBLE |
| WELDING | May 10, 2023 | HAMM & WITTKOPP | ADMISSIBLE |
| HANSEN | May 9, 2023 | MAIWALD | ADMISSIBLE |
| TEVA PHARMACEUTICALS | May 9, 2023 | KRAUS & LEDERER PARTGMBB | ADMISSIBLE |
| ELKINGTON AND FIFE | May 4, 2023 | ELKINGTON AND FIFE | ADMISSIBLE |
Patent citations refer to prior patents cited during different phases such as opposition or international search.
| Citation Phase | Publication Number |
|---|---|
| DESCRIPTION | US2004053908 |
| DESCRIPTION | US2007004773 |
| DESCRIPTION | US2007037849 |
| DESCRIPTION | US2007078159 |
| DESCRIPTION | US2007117842 |
| DESCRIPTION | WO2006030826 |
| DESCRIPTION | WO2011021597 |
| OPPOSITION | CN107305202 |
| OPPOSITION | EP1683785 |
| OPPOSITION | EP1698623 |
| OPPOSITION | EP1698923 |
| OPPOSITION | EP1777218 |
| OPPOSITION | EP1797881 |
| OPPOSITION | EP1894918 |
| OPPOSITION | EP3524595 |
| OPPOSITION | JP2014174062 |
| OPPOSITION | JP2015034729 |
| OPPOSITION | US2004053908 |
| OPPOSITION | US2007004773 |
| OPPOSITION | US2007037849 |
| OPPOSITION | US2007078159 |
| OPPOSITION | US2007117842 |
| OPPOSITION | US2008214604 |
| OPPOSITION | WO0232872 |
| OPPOSITION | WO2004101526 |
| OPPOSITION | WO2005044788 |
| OPPOSITION | WO2005063713 |
| OPPOSITION | WO2006030826 |
| OPPOSITION | WO2006137474 |
| SEARCH | EP1683785 |
| SEARCH | EP1698623 |
| SEARCH | EP1777218 |
| SEARCH | EP1797881 |
| SEARCH | EP1894918 |
| SEARCH | US2007117842 |
| SEARCH | WO0232872 |
| SEARCH | WO2004101526 |
| SEARCH | WO2005044788 |
| SEARCH | WO2005063713 |
| SEARCH | WO2006030826 |
| SEARCH | WO2006137474 |
The dossier documents provide a comprehensive record of the patent's prosecution history - including filings, correspondence, and decisions made by patent offices - and are crucial for understanding the patent's legal journey and any challenges it may have faced during examination.
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