Patent No. EP3524595 (titled "High-Purity Quinoline Derivative And Method For Manufacturing Same") was filed by Eisai R&D Management on Aug 26, 2015. The application was issued on Aug 10, 2022.
Quinline derivative that is easy to remove such impurities by a common purification method such as chromatography and crystallization. The derivative comprises a compound represented by formula (IV) or a salt thereof; an organometallic reagent such as butyllithium, methyllithium, lithium bistrimethylsilylamide, sodium bistrimethylsilylamide or potassium bistrimethylsilylamide; a hydride such as lithium hydride, sodium hydride or potassium hydride; a heterocyclic compound such as imidazole, pyridine, dimethylpyridine, trimethylpyridine or 4-dimethylaminopyridine; or an organic amine such as triethylamine, N,N-diisopropylethylamine or diazabicycloundecene.

Patent oppositions filed by competitors challenge the validity of a granted patent. These oppositions are typically based on claims of prior art, lack of novelty, or non-obviousness. They are a key part of the process for determining a patent's strength and enforceability.
| Company | Opposition Date | Representative |
|---|---|---|
| ACCORD HEALTHCARE | May 10, 2023 | UEXKULL & STOLBERG |
| AECHTER | May 10, 2023 | TER MEER STEINMEISTER & PARTNER |
| GENERICS UK | May 10, 2023 | RUSSELL |
| MAIWALD | May 10, 2023 | MAIWALD |
| STADA ARZNEIMITTEL | May 10, 2023 | HAMM & WITTKOPP |
| WELDING | May 10, 2023 | HAMM & WITTKOPP |
| HANSEN | May 9, 2023 | MAIWALD |
| TEVA PHARMACEUTICALS | May 9, 2023 | KRAUS & LEDERER PARTGMBB |
| ELKINGTON AND FIFE | May 4, 2023 | ELKINGTON AND FIFE |
The dossier documents provide a comprehensive record of the patent's prosecution history - including filings, correspondence, and decisions made by patent offices - and are crucial for understanding the patent's legal journey and any challenges it may have faced during examination.
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