Patent No. EP3666797 (titled "Antigen Binding Proteins To Proprotein Convertase Subtilisin Kexin Type 9 (Pcsk9)") was filed by Amgen on Aug 22, 2008. The application was issued on May 17, 2023.
Monoclonal antibodies that bind to the catalytic domain of PCSK9, a cholesterol-lowering protein, and prevent or reduce the binding of PCSK9 to LDLR. These antibodies can be used to treat or prevent hypercholesterolemia and atherosclerotic diseases by inhibiting PCSK9's function. The antibodies bind to specific regions of PCSK9's heavy and light chain variable domains.
Latest UPC cases involving this patent.
| Case Number | Filing Date | Plaintiff | Proceeding Type |
|---|---|---|---|
| UPC_CFI_0002221/2025 | Dec 23, 2025 | Amgen | Generic |
| UPC_CFI_0002220/2025 | Dec 23, 2025 | Amgen | Generic |
| APP_3214/2025 | Jan 21, 2025 | Name NOT Displayed FOR Gdpr Reasons Represented BY Sture Rygaard, Redacted Natural Person Name | Generic |
| UPC_COA_529/2024 | Sep 13, 2024 | Amgen | Appeal |
| UPC_COA_528/2024 | Sep 13, 2024 | Amgen | Appeal |
| APP_47172/2024 | Aug 14, 2024 | Dehns | Generic |
| APP_47163/2024 | Aug 14, 2024 | Dehns | Generic |
| APP_47154/2024 | Aug 14, 2024 | Dehns | Generic |
| CC_586764/2023 | Nov 10, 2023 | Regeneron Pharmaceuticals | Counter Claim For Revocation |
| APP_546231/2023 | Jul 11, 2023 | Name NOT Displayed FOR Gdpr Reasons Represented BY Oswin Ridderbusch, Redacted Natural Person Name | Generic |

Patent oppositions filed by competitors challenge the validity of a granted patent. These oppositions are typically based on claims of prior art, lack of novelty, or non-obviousness. They are a key part of the process for determining a patent's strength and enforceability.
| Company | Opposition Date | Representative |
|---|---|---|
| REGENERON PHARMACEUTICALS | Feb 19, 2024 | ZWICKER |
| SANOFI AVENTIS DEUTSCHLAND | Nov 10, 2023 | CARPMAELS & RANSFORD |
| SANOFI AVENTIS DEUTSCHLAND SANOFI AVENTIS GROUPE SANOFI WINTHROP INDUSTRIE | Nov 10, 2023 | CARPMAELS & RANSFORD |
The dossier documents provide a comprehensive record of the patent's prosecution history - including filings, correspondence, and decisions made by patent offices - and are crucial for understanding the patent's legal journey and any challenges it may have faced during examination.
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