Patent No. EP3756650 (titled "Formulations Of (+)-2-[1-(3-Ethoxy-4-Methoxy-Phenyl)-2-Methanesulfonyl-Ethyl]-4-Acetyl Aminoisoindoline-1,3-Dione") was filed by Amgen Europe on Dec 26, 2012. The application was issued on Aug 20, 2025.
Pharmaceutical compositions comprising (+)-2-[1-(3-ethoxy-4-methoxy-phenyl)-2-methanesulfonyl-ethyl]-4-acetylaminoisoindoline-1,3-dione (Compound A) for treating various diseases and disorders, including cancer, pain, inflammatory diseases, and ocular neovascular diseases. The compositions comprise Compound A in combination with fillers, disintegrants, and lubricants, and may be formulated as tablets or capsules. The compositions exhibit advantageous physical and pharmacological properties, including fast disintegration, low friability, and stability.

Patent oppositions filed by competitors challenge the validity of a granted patent. These oppositions are typically based on claims of prior art, lack of novelty, or non-obviousness. They are a key part of the process for determining a patent's strength and enforceability.
| Company | Opposition Date | Representative |
|---|---|---|
| COOKE | Mar 18, 2026 | ELKINGTON AND FIFE |
| BRAND MURRAY FULLER | Jan 12, 2026 | BRAND MURRAY FULLER |
| HAMM & WITTKOPP | Dec 19, 2025 | HAMM & WITTKOPP |
| TER MEER STEINMEISTER & PARTNER PATENTANWALTE MBB | Dec 8, 2025 | TER MEER STEINMEISTER & PARTNER |
| CAMULON | Oct 24, 2025 | REDDIE & GROSE |
| ELKINGTON AND FIFE | Oct 1, 2025 | ELKINGTON AND FIFE |
The dossier documents provide a comprehensive record of the patent's prosecution history - including filings, correspondence, and decisions made by patent offices - and are crucial for understanding the patent's legal journey and any challenges it may have faced during examination.
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